当前位置: 首页   >  成果及论文
成果及论文

Ge Xu, Bin-Hua Lv, Jacques Y. Roberge, Bai-Hua Xu, Ji-Yan Du, Jia-Jia Dong, Yuan-Wei Chen, Kun Peng, Li-Li Zhang, Xin-Xing Tang, Yan Feng, Min Xu, Wei Fu, Wen-Bin Zhang, Liang-Cheng Zhu, Zhong-Ping Deng, Ze-Lin Sheng, Ajith Welihinda, Xun Sun*. Design, synthesis, and biological evaluation of deuterated C-aryl glycoside as a potent and long-acting renal sodium-dependent glucose cotransporter 2 inhibitor for the treatment of type 2 diabetes. J. Med. Chem. 2014, 57, 1236-1251. (IF: 5.614) Cheng Xie, Jun Chang, Xiao-Dong Hao, Jian-Ming Yu, Hong-Rui Liu, Xun Sun*. Mitochondri-altargeted prodrug cancer therapy using a rhodamine B labeled fluorinated docetaxel. Eur. J. Pharm. Biopharm. 2013, 85, 541-549. (IF: 3.826) Chen Zhong, Xin-Hua Liu, Xiao-Dong Hao, Jun Chang, Xun Sun*. Synthesis and biological evaluation of novel neuroprotective agents for paraquat-induced apoptosis in human neuronal SH-SY5Y cells. Eur. J. Med. Chem. 2013, 62, 187–198. (IF: 3.499) Jun Chang, Si-Ji Zhang,Yong-Wei Jiang, Liang Xu, Jian-Ming Yu, Wen-Jiang Zhou, Xun Sun*. Design, synthesis and antibacterial activity of novel demethylvancomycin analogs against resistant bacteria. ChemMedChem. 2013, 8,976–984. (IF: 2.835) (封面文章) Chen Zhong, Xin-Hua Liu, Jun Chang, Jian-Ming Yu, Xun Sun*. Inhibitory effect of resveratrol dimerized derivatives on nitric oxide production in lipopolysaccharide-induced RAW 264.7 cells. Bioorg. Med. Chem. Lett. 2013, 23, 4413-4418. (IF: 2.338) Qing Yang, Jun Chang, Jiao Song, Meng-Ting Qian, Jian-Ming Yu, Xun Sun*. Synthesis and in vitro antitumor activity of novel iridium (III) complexes with enantiopure C2-symmetrical vicinal diamine ligands. Bioorg. Med. Chem. Lett. 2013. 23, 4602-4607. (IF: 2.338) Si-Ji Zhang, Qing Yang, Liang Xu, Jun Chang, Xun Sun*. Synthesis and antibacterial activity against Clostridium difficile of novel demethylvancomycin derivatives. Bioorg. Med. Chem. Lett. 2012, 22,4942–4945. (IF: 2.338) Hong-Fu Lu, Cheng Xie, Jun Chang, Guo-Qiang Lin, Xun Sun*. Synthesis, cytotoxicity, metabolic stability and pharmacokinetic evaluation of fluorinated docetaxel analogues. Eur. J. Med. Chem. 2011, 46, 1743-1748. (IF: 3.499) Chen Zhong, Jun Zhu, Jun Chang, Xun Sun*. Concise total syntheses of (±)isopaucifloral F, (±)quadrangularin A, and (±)pallidol. Tetrahedron Lett. 2011, 52, 2815–2817. (IF: 2.397) Hong-Fu Lu, Xun Sun*, Liang Xu, Li-Guang Lou, Guo-Qiang Lin. Design, synthesis and biological evaluation of novel fluorinated docetaxel analogues. Eur. J. Med. Chem. 2009, 44, 482-491. (IF: 3.499)